1 J3I (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(1-carbamimidoylpiperidin-4-yl)methyl]pyrrolidine-2-carboxamide 1.000 2 06P D-phenylalanyl-N-[(1-methylpyridinium-4-yl)methyl]-L-prolinamide 0.931 3 P05 D-phenylalanyl-N-(pyridin-4-ylmethyl)-L-prolinamide 0.897 4 M6Q (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(2-azanylpyridin-4-yl)methyl]pyrrolidine-2-carboxamide 0.867 5 GOZ (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[[2,6-bis(azanyl)pyridin-4-yl]methyl]pyrrolidine-2-carboxamide 0.839 6 53U D-phenylalanyl-N-benzyl-L-prolinamide 0.833 7 0BM N-(methylsulfonyl)-D-phenylalanyl-N-[(1-carbamimidoylpiperidin-4-yl)methyl]-L-prolinamide 0.824 8 22U D-phenylalanyl-N-(3-chlorobenzyl)-L-prolinamide 0.806 9 37U D-phenylalanyl-N-(3-fluorobenzyl)-L-prolinamide 0.806 10 51U D-phenylalanyl-N-(3-methylbenzyl)-L-prolinamide 0.806 11 64U 3-cyclohexyl-D-alanyl-N-(3-chlorobenzyl)-L-prolinamide 0.806 12 MD8 (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(4-hydroxyphenyl)methyl]pyrrolidine-2-carboxamide 0.806 13 K73 (2~{S})-~{N}-[[4-(aminomethyl)phenyl]methyl]-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]pyrrolidine-2-carboxamide 0.781 14 N6L D-phenylalanyl-N-(2,5-dichlorobenzyl)-L-prolinamide 0.781 15 99P D-phenylalanyl-N-(pyridin-3-ylmethyl)-L-prolinamide 0.774 16 32U D-phenylalanyl-N-{4-[amino(iminio)methyl]benzyl}-L-prolinamide 0.758 17 6OV 3-cyclohexyl-D-alanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 0.758 18 6TH (2~{S})-1-[(2~{R})-2-azanyl-3-cyclohexyl-propanoyl]-~{N}-[[5-chloranyl-2-(hydroxymethyl)phenyl]methyl]pyrrolidine-2-carboxamide 0.758 19 71U (2~{S})-~{N}-[[2-(aminomethyl)-5-chloranyl-phenyl]methyl]-1-[(2~{R})-2-azanyl-3-cyclohexyl-propanoyl]pyrrolidine-2-carboxamide 0.758 20 10P D-phenylalanyl-N-[(1-methylpyridinium-3-yl)methyl]-L-prolinamide 0.750 21 J5K (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(6-azanylpyridin-3-yl)methyl]pyrrolidine-2-carboxamide 0.750 22 P97 D-phenylalanyl-N-[(4-chloropyridin-3-yl)methyl]-L-prolinamide 0.750 23 LXW (2~{S})-1-[(2~{R})-2-azanyl-3,3-diphenyl-propanoyl]-~{N}-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide 0.743 24 27U N-(4-carbamimidoylbenzyl)-1-(3-phenylpropanoyl)-L-prolinamide 0.727 25 50U (S)-N-(4-carbamimidoylbenzyl)-1-(3-cyclohexylpropanoyl)pyrrolidine-2-carboxamide 0.727 26 98P D-phenylalanyl-N-[(4-chloro-1-methylpyridinium-3-yl)methyl]-L-prolinamide 0.727 27 MIN Methyl-phe-pro-amino-cyclohexylglycine 0.727 28 B03 D-phenylalanyl-N-(pyridin-2-ylmethyl)-L-prolinamide 0.719 29 MJK (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(5-bromanylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide 0.719 30 O5Z (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(5-bromanylfuran-2-yl)methyl]pyrrolidine-2-carboxamide 0.719 31 OQZ (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(5-chloranylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide 0.719 32 QKE (2~{S})-1-[(2~{R})-2-azanyl-3-phenyl-propanoyl]-~{N}-[(5-chloranylfuran-2-yl)methyl]pyrrolidine-2-carboxamide 0.719