1 IVK (3r,4r)-N-(4-chlorophenyl)-N'-[2-fluoro-4-(2-oxopyridin-1(2h)-yl)phenyl]-1-(2,2,2-trifluoroethyl)pyrrolidine-3,4-dicarboxamide 1.000 2 XBV (3r,4r)-1-(2,2-difluoro-ethyl)-pyrrolidine-3,4-dicarboxylic acid 3-[(5-chloro-pyridin-2-yl)-amide]-4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.921 3 63C (3r,4r)-1-methylcarbamoylmethyl-pyrrolidine-3,4-dicarboxylic acid 3-[(4-chloro-phenyl)-amide] 4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.850 4 455 (3r,4r)-1-sulfamoyl-pyrrolidine-3,4-dicarboxylic acid 3-[(4-chloro-phenyl)-amide] 4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.780 5 RR8 (3r,4r)-1-methanesulfonyl-pyrrolidine-3,4-dicarboxylic acid 3-[(4-chloro-phenyl)-amide] 4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.780 6 OYJ (3r,4r)-1-methanesulfonyl-pyrrolidine-3,4-dicarboxylic acid 3-[(4-chloro-3-fluoro-phenyl)-amide] 4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.762 7 8NC (3r,4r)-1-methanesulfonyl-pyrrolidine-3,4--dicarboxylic acid 3-[(3-fluoro-4-methoxy-phenyl)-amide] 4-{[2-fluoro-4-(2-oxo-2h-pyridin-1-yl)-phenyl]-amide} 0.705