1 I09 (3r,4r,5s)-3-(3-chlorophenyl)-4-(4-chlorophenyl)-4-cyano-N-[(3s)-3,4-dihydroxybutyl]-5-(2,2-dimethylpropyl)-D-prolinamide 1.000 2 1OY (3s,4r,5s)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-N-[(3s)-3,4-dihydroxybutyl]-5-(2,2-dimethylpropyl)-D-prolinamide 0.946 3 1MT (2'S,3r,4'S,5'R)-N-(2-aminoethyl)-6-chloro-4'-(3-chloro-2-fluorophenyl)-2'-(2,2-dimethylpropyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-5'-carboxamide 0.725