1 GVD [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile 1.000 2 IHH [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile 1.000 3 3RF N~2~-(4-aminophenyl)-N~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine 0.867 4 REB [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile 0.862 5 EBD [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrile 0.833 6 5CP [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile 0.806 7 38R [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile 0.750 8 3RJ N~2~-(1h-benzimidazol-6-yl)-N~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine 0.735