1 GS5 5-chloro-N-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-1-benzothiophene-2-sulfonamide 1.000 2 GS6 6-chloro-N-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-1-benzothiophene-2-sulfonamide 0.935 3 GSQ 5-chloro-N-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-5-chloro-N-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-sulfonamide 0.935 4 GSK 6-chloro-N-{(3s)-1-[(1s)-1-methyl-2-(4-morpholinyl)-2-oxo ethyl]-2-oxo-3-pyrrolidinyl}-2-naphthalenesulfonamide 0.848 5 GSX 5'-chloro-N-{(3s)-1-[(1s)-1-methyl-2-morpholin-4-yl-2-oxoethyl]-2-oxopyrrolidin-3-yl}-2,2'-bithiophene-5-sulfonamide 0.848 6 987 N-[(3s)-1-{(2s)-1-[(3s)-3-aminopiperidin-1-yl]-1-oxopropan-2-yl}-2-oxopyrrolidin-3-yl]-6-chloronaphthalene-2-sulfonamid E 0.771 7 4O4 6-chloro-N-{(3s)-1-[(2s)-1-(morpholin-4-yl)-1-oxopropan-2-yl]-2-oxo-2,3-dihydro-1h-pyrrol-3-yl}-N-(2-oxobutyl)naphthalene-2-sulfonamide 0.737 8 48W 6-chloro-N-{(3s)-1-[(2s)-1-(4-methyl-5-oxo-1,4-diazepan-1-yl)-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl}naphthalene-2-sulf onamide 0.730