1 FD3 N-alpha-(2-naphthylsulfonyl)-3-amidino-L-phenylalanine piperazide 1.000 2 FD4 N-alpha-(2-naphthylsulfonyl)-N(3-amidino-L-phenylalaninyl)-4-acetyl-piperazine 0.917 3 FD1 N-alpha-(2-naphthylsulfonyl)-N-(3-amidino-L-phenylalaninyl)-D-pipecolinic acid 0.865 4 FD2 N-alpha-(2-naphthylsulfonyl)-N(3-amidino-L-phenylalaninyl)isopipecolinic acid methyl ester 0.842 5 0N6 (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 0.829 6 1L4 N-[(2r)-3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-8-fluoro-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 0.806 7 0ZG 3-[(2s)-2-{[(4-methylphenyl)sulfonyl]amino}-3-oxo-3-piperidin-1-ylpropyl]benzenecarboximidamide 0.800 8 730 (S)-3-(3-(4-(2-guanidinoethyl)piperidin-1-yl)-2-(naphthalene-2-sulfonamido)-3-oxopropyl)benzimidamide 0.800 9 MUQ 4-[(2~{S})-3-(3-carbamimidoylphenyl)-2-[[3-(4-methoxy-2-oxidanyl-phenyl)phenyl]sulfonylamino]propanoyl]-~{N}-methyl-piperazine-1-carboxamide 0.744 10 0NW 3-[(2s)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-{[(2',4'-dichlorobiphenyl-3-yl)sulfonyl]amino}-3-oxopropyl]benzenecarboximidamide 0.738 11 1L8 8-fluoro-N-{(2r)-1-oxo-1-(pyrrolidin-1-yl)-3-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 0.718