1 CRV N-[1-(aminomethyl)cyclopropyl]-3-(benzylsulfonyl)-N~2~-[(1s)-2,2,2-trifluoro-1-(4-hydroxyphenyl)ethyl]-L-alaninamide 1.000 2 CRJ N-(1-cyanocyclopropyl)-3-({[(2s)-5-oxopyrrolidin-2-yl]methyl}sulfonyl)-N~2~-[(1s)-2,2,2-trifluoro-1-(4-fluorophenyl)ethyl]-L-alaninamide 0.833