1 CO4 2,4-diamino-5-methyl-6-[(3,4,5-trimethoxy-N-methylanilino)methyl]pyrido[2,3-D]pyrimidine 1.000 2 TMQ Trimetrexate 0.897 3 TQD (2r,6s)-6-{[methyl(3,4,5-trimethoxyphenyl)amino]methyl}-1,2,5,6,7,8-hexahydroquinazoline-2,4-diamine 0.897 4 VG9 6-{[(2,5-diethoxyphenyl)amino]methyl}-5-methylpyrido[2,3-D]pyrimidine-2,4-diamine 0.719