1 C1P N~2~-(morpholin-4-ylcarbonyl)-N-[(3s)-1-phenyl-5-(phenylsulfonyl)pentan-3-yl]-L-leucinamide 1.000 2 0D6 N-{(1r)-3-phenyl-1-[2-(phenylsulfonyl)ethyl]propyl}-N~2~-(piperazin-1-ylcarbonyl)-L-leucinamide 0.947 3 4MC (z)-N-(5-guanidino-1-oxo-1-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-ylamino)pentan-2-yl)-4-methylpiperazine-1-carboxamid E 0.814 4 2V5 N-[(2s)-5-(carbamimidamidooxy)-1-oxo-1-{[(1e,3s)-5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl]amino}pentan-2-yl]-4-methylpiperazine-1-carboxamide 0.795 5 VS1 3-[[N-[morpholin-N-yl]-carbonyl]-phenylalaninyl-amino]-5- phenyl-pentane-1-sulfonylbenzene 0.791 6 MQQ N-[(1s)-1-[({(1s)-3-phenyl-1-[2-(phenylsulfonyl)ethyl]propyl}amino)carbonyl]-3-(phenylsulfonyl)propyl]morpholine-4-carboxamide 0.761 7 0IW Nalpha-[(4-methylpiperazin-1-yl)carbonyl]-N-[(3s)-1-phenyl-5-(phenylsulfonyl)pentan-3-yl]-L-phenylalaninamide 0.733 8 D1R Nalpha-[(4-methylpiperazin-1-yl)carbonyl]-N-{(1s)-3-phenyl-1-[2-(phenylsulfonyl)ethyl]propyl}-L-phenylalaninamide 0.733 9 0I5 N-[(3s)-1-fluoro-2-oxo-5-phenylpentan-3-yl]-N~2~-(morpholin-4-ylcarbonyl)-L-leucinamide 0.718 10 BCQ N-[(1r)-1-[({[(5s)-3,5-dimethyl-2,5-dihydroisoxazol-4-yl]methyl}sulfonyl)methyl]-2-oxo-2-({(1s)-3-phenyl-1-[2-(phenylsulfonyl)ethyl]propyl}amino)ethyl]morpholine-4-carboxamide 0.708