1 BJS 2-(3-[3-({3-[(benzylamino)methyl]-4-chlorophenyl}ethynyl)-4-chlorophenyl]-1-{3-[(3s)-3-methylmorpholin-4-yl]propyl}-1,4,6,7-tetrahydro-5h-pyrazolo[4,3-C]pyridin-5-yl)-2-oxoacetamide 1.000 2 BJD N-benzyl-1-{2-chloro-5-[(2-chloro-5-{5-(methylsulfonyl)-1-[3-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1h-pyrazolo[4,3-C]pyridin-3-yl}phenyl)ethynyl]phenyl}methanamine 0.811 3 BJJ N-benzyl-1-{2-chloro-5-[2-(2-chloro-5-{5-(methylsulfonyl)-1-[3-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1h-pyrazolo[4,3-C]pyridin-3-yl}phenyl)ethyl]phenyl}methanamine 0.811 4 BFV N-benzyl-1-{3-[(2-chloro-5-{5-(methylsulfonyl)-1-[3-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1h-pyrazolo[4,3-C]pyridin-3-yl}phenyl)ethynyl]phenyl}methanamine 0.792 5 599 2-[3-{4-chloro-3-[(4-chlorophenyl)ethynyl]phenyl}-1-(3-morpholin-4-ylpropyl)-1,4,6,7-tetrahydro-5h-pyrazolo[4,3-C]pyridin-5-yl]-2-oxoethanol 0.776 6 BJV N-benzyl-1-{5-[(2-chloro-5-{5-(methylsulfonyl)-1-[3-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1h-pyrazolo[4,3-C]pyridin-3-yl}phenyl)ethynyl]-2-methoxyphenyl}methanamine 0.764