1 AE8 (S)-4-((4-(((2,3-dihydro-[1,4]dioxino[2,3-C]pyridin-7-yl)methyl)amino)piperidin-1-yl)methyl)-3-fluoro-4-hydroxy-4h-pyrrolo[3,2,1-de][1,5]naphthyridin-7(5h)-one 1.000 2 6EJ (1r)-1-[(4-{[(6,7-dihydro[1,4]dioxino[2,3-C]pyridazin-3-yl)methyl]amino}piperidin-1-yl)methyl]-9-fluoro-1,2-dihydro-4h-pyrrolo[3,2,1-ij]quinolin-4-one 0.861 3 JHN (3~{R})-3-[[4-(3,4-dihydro-2~{H}-pyrano[2,3-C]pyridin-6-ylmethylamino)piperidin-1-yl]methyl]-1,4,7-triazatricyclo[6.3.1.0^{4,12}]dodeca-6,8(12),9-triene-5,11-dione 0.811