1 A61 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzothiazol-6-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 1.000 2 K19 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzothiazol-6-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.976 3 XUY (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.952 4 A60 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl](2-ethylbutyl)amino}-1-benzyl-2-hydroxypropyl]carbamate 0.907 5 F53 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-3-[(2-ethylbutyl){[4-(hydroxymethyl)phenyl]sulfonyl}amino]-2-hydroxypropyl}carbamate 0.886 6 K2D (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-3-{(2-ethylbutyl)[(4-methoxyphenyl)sulfonyl]amino}-2-hydroxypropyl]carbamate 0.886 7 K13 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl][(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.884 8 K2E (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzodioxol-5-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.867 9 NF4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[(2-ethylbutyl)({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.867 10 NFJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[(2-ethylbutyl)({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.867 11 K14 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl][(2s)-2-methylbutyl]amino}propyl]carbamate 0.864 12 K2A (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-({[4-(hydroxymethyl)phenyl]sulfonyl}[(2s)-2-methylbutyl]amino)propyl]carbamate 0.864 13 017 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(1s,2r)-3-[[(4-aminophenyl)sulfonyl](isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate 0.860 14 C7U (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.848 15 NJ1 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-ethylbutyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.848 16 NJJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-ethylbutyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.848 17 YUA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{(2-ethylbutyl)[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.848 18 K20 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzodioxol-5-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.844 19 NE7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.844 20 NEJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.844 21 C7J (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.841 22 DJR (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}propyl]carbamate 0.841 23 NJM (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[4-(hydroxymethyl)phenyl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.841 24 P3V (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3,3-dihydroxy-1-phenylbutan-2-yl]carbamate 0.841 25 NJ7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.826 26 NJG (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.826 27 YUD (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl][(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.826 28 065 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(2s,3r)-3-hydroxy-4-(N-isobutylbenzo[D][1,3]dioxole-5-sulfonamido)-1-phenylbutan-2-ylcarbamate 0.822 29 4UX (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.822 30 BVR [4-[[(2~{R},3~{S})-3-[[(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl]oxycarbonylamino]-2-oxidanyl-4-phenyl-butyl]-(2-methylpropyl)sulfamoyl]phenyl]-oxidanyl-oxidanylidene-boron 0.822 31 G07 4-{[(2r,3s)-3-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-2-hydroxy-4-phenylbutyl](2-methylpropyl)sulfamoyl}benzoic acid 0.822 32 G08 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-carbamoylphenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.822 33 G10 (3r,3as,6as)-4,4-difluorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.822 34 NJ4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.822 35 NJA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.822 36 0TQ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({(3z)-3-[1-(methylamino)ethylidene]-2-oxo-2,3-dihydro-1h-indol-5-yl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.812 37 XVV Diethyl [(4-{(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-ethylbutyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.808 38 4UY (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.804 39 G04 (3r,3as,4r,6ar)-4-methoxyhexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.804 40 NF7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.804 41 NG4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.804 42 YUJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.804 43 7O7 (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.796 44 G8R (1r,3as,4s,6s,7ar)-octahydro-1,6-epoxy-2-benzofuran-4-yl [(2s,3r)-4-{[2-(cyclopropylamino)-1,3-benzothiazole-6-sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.796 45 QK1 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl {(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzothiazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.796 46 478 {3-[(4-amino-benzenesulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxy-propyl}-carbamic acid tetrahydro-furan-3-yl ester 0.791 47 XVJ Diethyl [(4-{(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl][(2s)-2-methylbutyl]amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.788 48 G43 [(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl] ~{N}-[(2~{S},3~{R})-1-(3-chloranyl-4-methoxy-phenyl)-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-butan-2-yl]carbamate 0.787 49 G52 (3r,3as,3br,6as,7as)-octahydrodifuro[2,3-B:3',2'-D]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.787 50 X7H (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[4-(2-chloroacetamido)benzene-1-sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.787 51 YUP (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-[{4-[(1s)-1-hydroxyethyl]benzene-1-sulfonyl}(2-methylpropyl)amino]butan-2-yl}carbamate 0.787 52 52U (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.783 53 QHA (3r,3as,4r,6ar)-4-[(2-fluoroprop-2-en-1-yl)oxy]hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.780 54 QJY (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl {(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzothiazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.780 55 ZLP (3r,3as,4r,6ar)-4-(2-methoxyethoxy)hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[(2z)-2-(methylimino)-2,3-dihydro-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.780 56 G55 (5r)-1,3-dioxepan-5-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.778 57 6KK (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-[(3r,5r,7r)-tricyclo[3.3.1.1~3,7~]decan-1-yl]butan-2-yl}carbamate 0.771 58 C7L (3r,3as,4r,6ar)-4-(2-methoxyethoxy)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.771 59 X7B [(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl] ~{N}-[(2~{S},3~{R})-4-[[7,7-bis(oxidanyl)-9-oxidanylidene-8-oxa-7-boranuidabicyclo[4.3.0]nona-1,3,5-trien-3-yl]sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-1-phenyl-butan-2-yl]carbamate 0.771 60 XUP Diethyl [(4-{(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-methylpropyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.769 61 52W (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.766 62 8FM (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.766 63 B4R {4-[{(2r,3s)-3-[({[(3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}boronic acid 0.766 64 FQ4 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.766 65 T1R (1r,3as,5r,6s,7ar)-octahydro-1,6-epoxy-2-benzofuran-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.766 66 G77 (1s,3ar,4r,6r,7as)-octahydro-1,6-epoxy-2-benzofuran-4-yl [(2s,3r)-4-{[2-(cyclopropylamino)-1,3-benzothiazole-6-sulfonyl](2-methylpropyl)amino}-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.765 67 J5L (3r,3as,4r,6ar)-4-[2-(methylamino)-2-oxoethoxy]hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[(2z)-2-(methylimino)-2,3-dihydro-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.765 68 GRL (3as,5r,6ar)-hexahydro-2h-cyclopenta[B]furan-5-yl (2s,3s)-3-hydroxy-4-(4-(hydroxymethyl)-N-isobutylphenylsulfonamido)-1-phenylbutan-2-ylcarbamate 0.761 69 T2R (1s,3ar,5s,6r,7as)-octahydro-1,6-epoxy-2-benzofuran-5-yl {(2s,3r)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]-1-phenylbutan-2-yl}carbamate 0.760 70 GR6 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-2-hydroxy-3-[(7e)-13-methoxy-1,1-dioxido-3,4,5,6,9,10-hexahydro-2h-11,1,2-benzoxathiazacyclotridecin-2-yl]propyl}carbamate 0.755 71 GR7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[(7e)-13-methoxy-1,1-dioxo-1,4,5,6,9,11-hexahydro-10,1lambda~6~,2-benzoxathiazacyclotridecin-2(3h)-yl]-1-phenylbutan-2-yl}carbamate 0.755 72 53F (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-(4-methoxyphenyl)butan-2-yl]carbamate 0.750 73 5B7 (3r,3ar,4s,7as)-3-methoxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.750 74 C7W (3r,3as,4r,6ar)-4-(3,3,3-trifluoropropoxy)hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.750 75 FQ1 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.750 76 Q1D {4-[{(2r,3s)-3-[({[(3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}boronic acid 0.750 77 G05 (4ar,6r,7as)-hexahydro-4ah-cyclopenta[B][1,4]dioxin-6-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.745 78 G89 (3r,3ar,5r,6ar)-3-hydroxyhexahydro-2h-cyclopenta[B]furan-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.745 79 J0S (3as,5r,6ar)-2-oxohexahydro-2h-cyclopenta[D][1,3]oxazol-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.745 80 JDV (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(4-fluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.745 81 JDY (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3-fluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.745 82 74T (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({2-[(1-cyclopentylpiperidin-4-yl)amino]-1,3-benzothiazol-6-yl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-P henylbutan-2-yl}carbamate 0.741 83 QFI ({4-[(2s,3r)-2-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-3-hydroxy-4-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}butyl]phenoxy}methyl)phosphonic acid 0.740 84 VXL (3r,3as,4r,6ar)-4-[2-(methylamino)-2-oxoethoxy]hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.740 85 TK7 Diethyl [(4-{(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-ethylbutyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.736 86 52Z (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-1-(4-methoxyphenyl)-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.735 87 5B5 (3r,3as,4s,7as)-3-(ethylamino)hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.735 88 G79 (3ar,3br,4s,7ar,8as)-decahydrofuro[2,3-B][1]benzofuran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.735 89 7OA (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.731 90 G53 Methyl 2-{4-[{(2r,3s)-3-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}-1,3-oxazole-4-carboxylate 0.725 91 XVS Diethyl [(4-{(2s,3r)-4-{(2-ethylbutyl)[(4-methoxyphenyl)sulfonyl]amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.722 92 XVY Diethyl [(4-{(2s,3r)-4-[(2-ethylbutyl){[4-(hydroxymethyl)phenyl]sulfonyl}amino]-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.722 93 6KR (3r,3as,7ar)-hexahydro-4h-furo[2,3-B]pyran-3-yl {(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-[(3r,5r,7r)-tricyclo[3.3.1.1~3,7~]decan-1-yl]butan-2-yl}carbamate 0.720 94 GR5 (2ar,4s,4ar,7ar,7br)-octahydro-2h-1,7-dioxacyclopenta[Cd]inden-4-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.717 95 GR8 (2as,4r,4as,7as,7bs)-octahydro-2h-1,7-dioxacyclopenta[Cd]inden-4-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.717 96 XUS Diethyl [(4-{(2s,3r)-4-{[(4-aminophenyl)sulfonyl][(2s)-2-methylbutyl]amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.717 97 NJY (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-1-(3-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.712 98 NKA (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.712 99 XW4 Diethyl [(4-{(2s,3r)-4-{[(2h-1,3-benzodioxol-5-yl)sulfonyl](2-ethylbutyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.709 100 YTY Diethyl [(4-{(2s,3r)-4-[(2-ethylbutyl){4-[(1s)-1-hydroxyethyl]benzene-1-sulfonyl}amino]-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.709 101 XUV Diethyl ({4-[(2s,3r)-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl][(2s)-2-methylbutyl]amino}butyl]phenoxy}methyl)phosphonate 0.704 102 XVP Diethyl ({4-[(2s,3r)-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxy-4-({[4-(hydroxymethyl)phenyl]sulfonyl}[(2s)-2-methylbutyl]amino)butyl]phenoxy}methyl)phosphonate 0.704