1 92M 9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-B][1,4]diazepin -6(7h)-one 1.000 2 4WG 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-B][1,4]benzodiazepin-6-one 0.816 3 ZTX 2-((4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5,11-dimethyl-5h-benzo[E]pyrimido [5,4-B][1,4]diazepin-6(11h)-one 0.784 4 X7Y 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-B][1,4]benzodiazepin-6-one 0.744 5 X8J 5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-B][1,4]benzodiazepin-6-one 0.725