1 89D 17-{[ethyl(dihydroxy)-lambda~4~-sulfanyl]amino}-11,13-difluoro-2-methyl-6,7,8,9-tetrahydrodibenzo[4,5:7,8][1,6]dioxacyclododecino[3,2-C]pyridin-3(2h)-one 1.000 2 88M 5-[2-(2,4-difluorophenoxy)-5-{[ethyl(dihydroxy)-lambda~4~-sulfanyl]amino}phenyl]-4-ethoxy-1-methylpyridin-2(1h)-one 0.941 3 87D N-[3-(4-methoxy-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-4-phenoxyphenyl]methanesulfonamide 0.824 4 8NG N-[4-(2,4-difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1h-pyrrolo[2,3-C]pyridin-4-yl)phenyl]ethanesulfonamide 0.784 5 8NM N-[3-(6-methyl-7-oxo-6,7-dihydro-1h-pyrrolo[2,3-C]pyridin-4-yl)-4-phenoxyphenyl]methanesulfonamide 0.703