1 6KR (3r,3as,7ar)-hexahydro-4h-furo[2,3-B]pyran-3-yl {(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-[(3r,5r,7r)-tricyclo[3.3.1.1~3,7~]decan-1-yl]butan-2-yl}carbamate 1.000 2 6KK (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-[(3r,5r,7r)-tricyclo[3.3.1.1~3,7~]decan-1-yl]butan-2-yl}carbamate 0.933 3 DJR (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}propyl]carbamate 0.844 4 G52 (3r,3as,3br,6as,7as)-octahydrodifuro[2,3-B:3',2'-D]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.830 5 52U (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.826 6 G05 (4ar,6r,7as)-hexahydro-4ah-cyclopenta[B][1,4]dioxin-6-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.826 7 G89 (3r,3ar,5r,6ar)-3-hydroxyhexahydro-2h-cyclopenta[B]furan-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.826 8 K14 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl][(2s)-2-methylbutyl]amino}propyl]carbamate 0.826 9 G55 (5r)-1,3-dioxepan-5-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.822 10 4UY (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.809 11 52W (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.809 12 8FM (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.809 13 FQ4 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.809 14 G04 (3r,3as,4r,6ar)-4-methoxyhexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.809 15 K2D (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-3-{(2-ethylbutyl)[(4-methoxyphenyl)sulfonyl]amino}-2-hydroxypropyl]carbamate 0.809 16 T1R (1r,3as,5r,6s,7ar)-octahydro-1,6-epoxy-2-benzofuran-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.809 17 5B7 (3r,3ar,4s,7as)-3-methoxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.792 18 FQ1 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.792 19 G43 [(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl] ~{N}-[(2~{S},3~{R})-1-(3-chloranyl-4-methoxy-phenyl)-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-butan-2-yl]carbamate 0.792 20 J0S (3as,5r,6ar)-2-oxohexahydro-2h-cyclopenta[D][1,3]oxazol-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.787 21 017 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(1s,2r)-3-[[(4-aminophenyl)sulfonyl](isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate 0.783 22 52Z (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-1-(4-methoxyphenyl)-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.776 23 5B5 (3r,3as,4s,7as)-3-(ethylamino)hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.776 24 G79 (3ar,3br,4s,7ar,8as)-decahydrofuro[2,3-B][1]benzofuran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.776 25 C7J (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.766 26 GRL (3as,5r,6ar)-hexahydro-2h-cyclopenta[B]furan-5-yl (2s,3s)-3-hydroxy-4-(4-(hydroxymethyl)-N-isobutylphenylsulfonamido)-1-phenylbutan-2-ylcarbamate 0.766 27 K13 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl][(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.766 28 NJM (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[4-(hydroxymethyl)phenyl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.766 29 P3V (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3,3-dihydroxy-1-phenylbutan-2-yl]carbamate 0.766 30 6KQ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-{benzyl[(4-methoxyphenyl)sulfonyl]amino}-3-hydroxy-1-[(3r,5r,7r)-tricyclo[3.3.1.1~3,7~]decan-1-yl]butan-2-yl}carbamate 0.765 31 0JV Methyl N-[(3s,3ar,5r,6ar)-5-[[(2s,3r)-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-1-phenyl-butan-2-yl]carbamoyloxy]-3,3a,4,5,6,6a-hexahydro-2h-cyclopenta[B]furan-3-yl]carbamate 0.760 32 478 {3-[(4-amino-benzenesulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxy-propyl}-carbamic acid tetrahydro-furan-3-yl ester 0.756 33 065 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(2s,3r)-3-hydroxy-4-(N-isobutylbenzo[D][1,3]dioxole-5-sulfonamido)-1-phenylbutan-2-ylcarbamate 0.750 34 4UX (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.750 35 A60 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl](2-ethylbutyl)amino}-1-benzyl-2-hydroxypropyl]carbamate 0.750 36 BVR [4-[[(2~{R},3~{S})-3-[[(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl]oxycarbonylamino]-2-oxidanyl-4-phenyl-butyl]-(2-methylpropyl)sulfamoyl]phenyl]-oxidanyl-oxidanylidene-boron 0.750 37 G07 4-{[(2r,3s)-3-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-2-hydroxy-4-phenylbutyl](2-methylpropyl)sulfamoyl}benzoic acid 0.750 38 G08 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-carbamoylphenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.750 39 G10 (3r,3as,6as)-4,4-difluorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.750 40 K2A (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-({[4-(hydroxymethyl)phenyl]sulfonyl}[(2s)-2-methylbutyl]amino)propyl]carbamate 0.750 41 NJ4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.750 42 NJA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.750 43 XUY (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.750 44 QFI ({4-[(2s,3r)-2-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-3-hydroxy-4-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}butyl]phenoxy}methyl)phosphonic acid 0.745 45 VXL (3r,3as,4r,6ar)-4-[2-(methylamino)-2-oxoethoxy]hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.745 46 B4R {4-[{(2r,3s)-3-[({[(3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}boronic acid 0.735 47 F53 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-3-[(2-ethylbutyl){[4-(hydroxymethyl)phenyl]sulfonyl}amino]-2-hydroxypropyl}carbamate 0.735 48 K19 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzothiazol-6-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.735 49 K20 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzodioxol-5-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.735 50 NE7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.735 51 NEJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.735 52 NF7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.735 53 NG4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.735 54 YUJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.735 55 GR6 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-2-hydroxy-3-[(7e)-13-methoxy-1,1-dioxido-3,4,5,6,9,10-hexahydro-2h-11,1,2-benzoxathiazacyclotridecin-2-yl]propyl}carbamate 0.725 56 GR7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[(7e)-13-methoxy-1,1-dioxo-1,4,5,6,9,11-hexahydro-10,1lambda~6~,2-benzoxathiazacyclotridecin-2(3h)-yl]-1-phenylbutan-2-yl}carbamate 0.725 57 53F (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-(4-methoxyphenyl)butan-2-yl]carbamate 0.720 58 A61 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzothiazol-6-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.720 59 K2E (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzodioxol-5-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.720 60 NF4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[(2-ethylbutyl)({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.720 61 NFJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[(2-ethylbutyl)({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.720 62 NJ7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 63 NJG (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 64 Q1D {4-[{(2r,3s)-3-[({[(3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}boronic acid 0.720 65 X7H (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[4-(2-chloroacetamido)benzene-1-sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 66 YUD (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl][(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.720 67 YUP (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-[{4-[(1s)-1-hydroxyethyl]benzene-1-sulfonyl}(2-methylpropyl)amino]butan-2-yl}carbamate 0.720 68 C7L (3r,3as,4r,6ar)-4-(2-methoxyethoxy)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.706 69 C7U (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.706 70 NJ1 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-ethylbutyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.706 71 NJJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-ethylbutyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.706 72 X7B [(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl] ~{N}-[(2~{S},3~{R})-4-[[7,7-bis(oxidanyl)-9-oxidanylidene-8-oxa-7-boranuidabicyclo[4.3.0]nona-1,3,5-trien-3-yl]sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-1-phenyl-butan-2-yl]carbamate 0.706 73 YUA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{(2-ethylbutyl)[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl]amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.706