1 5MF 8-ethyl-5-methyl-2-[2-(2-methyl-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl)ethyl]-[1,2,4]triazolo[1,5-C]pyrimidine 1.000 2 IFR (4r)-5,7,8-trimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-C]pyrimidine 0.923 3 IQF (4r)-5-ethyl-8-methyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-C]pyrimidine 0.923 4 JTX (4s)-5-methyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}-8-(trifluoromethyl)[1,2,4]triazolo[1,5-C]pyrimidine 0.857 5 5M9 6-chloranyl-5,8-dimethyl-2-[2-(2-methyl-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl)ethyl]-[1,2,4]triazolo[1,5-a]pyridine 0.852 6 JIV (4s)-8-chloro-5,7-dimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-C]pyrimidine 0.852 7 K2L 1-(2-{2-[(4s)-5,8-dimethyl[1,2,4]triazolo[1,5-C]pyrimidin-2-yl]ethyl}-1-methyl-1h-imidazol-4-yl)pyrrolidin-2-one 0.852 8 IZH (4s)-5,8-dimethyl-2-(2-{1-methyl-3-[(2r)-2-(trifluoromethyl)pyrrolidin-1-yl]-1h-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-C]pyrimidine 0.828 9 IVT (4s)-5,8-dimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine 0.815 10 IGO (4s)-5,6,8-trimethyl-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine 0.786 11 IKU (4s)-5,8-dimethyl-2-(2-{1-methyl-3-[(2s)-2-methylpyrrolidin-1-yl]-1h-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-a]pyrazine 0.786 12 IOU (4s)-5,8-dimethyl-2-(2-{1-methyl-3-[(3s)-3-methylpyrrolidin-1-yl]-1h-1,2,4-triazol-5-yl}ethyl)[1,2,4]triazolo[1,5-a]pyrazine 0.786 13 JAP (4s)-2-(2-{3-[(3r)-3-fluoropyrrolidin-1-yl]-1-methyl-1h-1,2,4-triazol-5-yl}ethyl)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazine 0.786 14 IFE (4r)-6-chloro-2-{(E)-2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethenyl}[1,2,4]triazolo[1,5-a]pyridine 0.778 15 IFV (4r)-6-chloro-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyridine 0.778 16 IOZ (4s)-5,8-dimethyl-2-{2-[1-methyl-5-(pyrrolidin-1-yl)-1h-1,2,4-triazol-3-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine 0.750 17 JBV (4s)-2-(2-{3-[(3s)-3-(difluoromethyl)pyrrolidin-1-yl]-1-methyl-1h-1,2,4-triazol-5-yl}ethyl)-5,8-dimethyl[1,2,4]triazolo[1,5-a]pyrazine 0.733 18 IKB (4s)-5,8-dimethyl-2-{2-[1-methyl-3-(piperidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]pyrazine 0.724 19 IHL (4r)-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}-6-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyridine 0.700 20 IV8 (10r)-2-{2-[1-methyl-3-(pyrrolidin-1-yl)-1h-1,2,4-triazol-5-yl]ethyl}[1,2,4]triazolo[1,5-a]quinoline 0.700