1 5BP N-cyclopropyl-4-pyrazolo[1,5-B]pyridazin-3-ylpyrimidin-2-amine 1.000 2 KQW ~{N}-cyclopropyl-~{N}-methyl-4-pyrazolo[1,5-B]pyridazin-3-yl-pyrimidin-2-amine 0.950 3 KRQ ~{N}-methyl-4-pyrazolo[1,5-B]pyridazin-3-yl-pyrimidin-2-amine 0.800 4 KQK ~{N},~{N}-dimethyl-4-pyrazolo[1,5-B]pyridazin-3-yl-pyrimidin-2-amine 0.762 5 KR8 ~{N}-methyl-~{N}-phenyl-4-pyrazolo[1,5-B]pyridazin-3-yl-pyrimidin-2-amine 0.750