1 4T6 N~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-N~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine 1.000 2 4T5 N~2~-[(trans-4-aminocyclohexyl)methyl]-N~4~-(3-cyclopropyl-1h-pyrazol-5-yl)pyrimidine-2,4-diamine 0.821 3 C7Y N~4~-(5-cyclopropyl-1h-pyrazol-3-yl)-N~2~-[(1s)-1-(1h-pyrrolo[3,2-B]pyridin-5-yl)ethyl]pyrimidine-2,4-diamine 0.800 4 39I ~{N}4-(3-cyclopropyl-1~{H}-pyrazol-5-yl)-~{N}2-(phenylmethyl)thieno[3,2-D]pyrimidine-2,4-diamine 0.767