1 4RY N-[(4as,6s,8ar)-2-amino-5,6,7,8-tetrahydro-4a,8a-(methanooxymethano)-3,1-benzothiazin-6(4h)-yl]-3-chlorobenzamide 1.000 2 4RX N-[(4s,4as,6s,8ar)-10-aminohexahydro-3h-4,8a-(epithiomethenoazeno)isochromen-6(1h)-yl]-3-chlorobenzamide 0.920 3 4RZ N-[(4as,6s,8ar)-2-amino-4a,5,6,7,8,8a-hexahydro-4h-3,1-benzothiazin-6-yl]-3-chlorobenzamide 0.875 4 LWD ~{N}-quinolin-6-ylbenzamide 0.720 5 3YS N-{3-[(4as,7as)-2-amino-4a,5-dihydro-4h-furo[3,4-D][1,3]thiazin-7a(7h)-yl]-4-fluorophenyl}-5-fluoropyridine-2-carboxamide 0.700