1 385 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-[(1,3-benzodioxol-5-ylsulfonyl)(isobutyl)amino]-2-hydroxy-1-{4-[(2-methyl-1,3-thiazol-4-yl)methoxy]benzyl}propyl]carbamate 1.000 2 YUM (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-[{4-[(1s)-1-hydroxyethyl]benzene-1-sulfonyl}(2-methylpropyl)amino]-1-{4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl}butan-2-yl]carbamate 0.882 3 065 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(2s,3r)-3-hydroxy-4-(N-isobutylbenzo[D][1,3]dioxole-5-sulfonamido)-1-phenylbutan-2-ylcarbamate 0.833 4 K20 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzodioxol-5-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.816 5 K2E (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzodioxol-5-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.800 6 G43 [(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl] ~{N}-[(2~{S},3~{R})-1-(3-chloranyl-4-methoxy-phenyl)-4-[(4-methoxyphenyl)sulfonyl-(2-methylpropyl)amino]-3-oxidanyl-butan-2-yl]carbamate 0.765 7 017 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(1s,2r)-3-[[(4-aminophenyl)sulfonyl](isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate 0.755 8 C7U (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.750 9 XUM Diethyl [(4-{(2s,3r)-4-{[(2h-1,3-benzodioxol-5-yl)sulfonyl](2-methylpropyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.750 10 C7J (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.740 11 DJR (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}propyl]carbamate 0.740 12 K13 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl][(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.740 13 NJM (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[4-(hydroxymethyl)phenyl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.740 14 P3V (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3,3-dihydroxy-1-phenylbutan-2-yl]carbamate 0.740 15 XVM Diethyl [(4-{(2s,3r)-4-{[(2h-1,3-benzodioxol-5-yl)sulfonyl][(2s)-2-methylbutyl]amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.737 16 53F (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-(4-methoxyphenyl)butan-2-yl]carbamate 0.731 17 4UX (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.725 18 A60 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl](2-ethylbutyl)amino}-1-benzyl-2-hydroxypropyl]carbamate 0.725 19 BVR [4-[[(2~{R},3~{S})-3-[[(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl]oxycarbonylamino]-2-oxidanyl-4-phenyl-butyl]-(2-methylpropyl)sulfamoyl]phenyl]-oxidanyl-oxidanylidene-boron 0.725 20 G07 4-{[(2r,3s)-3-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-2-hydroxy-4-phenylbutyl](2-methylpropyl)sulfamoyl}benzoic acid 0.725 21 G08 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-carbamoylphenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.725 22 G10 (3r,3as,6as)-4,4-difluorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.725 23 K14 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl][(2s)-2-methylbutyl]amino}propyl]carbamate 0.725 24 K2A (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-({[4-(hydroxymethyl)phenyl]sulfonyl}[(2s)-2-methylbutyl]amino)propyl]carbamate 0.725 25 NJ4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.725 26 NJA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.725 27 XUY (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.725 28 XW4 Diethyl [(4-{(2s,3r)-4-{[(2h-1,3-benzodioxol-5-yl)sulfonyl](2-ethylbutyl)amino}-2-[({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl]oxy}carbonyl)amino]-3-hydroxybutyl}phenoxy)methyl]phosphonate 0.724 29 QFI ({4-[(2s,3r)-2-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-3-hydroxy-4-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}butyl]phenoxy}methyl)phosphonic acid 0.722 30 52Z (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-1-(4-methoxyphenyl)-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.717 31 4UY (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.712 32 F53 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-3-[(2-ethylbutyl){[4-(hydroxymethyl)phenyl]sulfonyl}amino]-2-hydroxypropyl}carbamate 0.712 33 G04 (3r,3as,4r,6ar)-4-methoxyhexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.712 34 K19 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzothiazol-6-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.712 35 K2D (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-3-{(2-ethylbutyl)[(4-methoxyphenyl)sulfonyl]amino}-2-hydroxypropyl]carbamate 0.712 36 NE7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.712 37 NEJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.712 38 NF7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.712 39 NG4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.712 40 YUJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.712