1 2LI N-[(1s,2r)-3-{[(5s)-5-(3-tert-butylphenyl)-4,5,6,7-tetrahydro-1h-indazol-5-yl]amino}-1-(3,5-difluorobenzyl)-2-hydroxypropyl]acetamide 1.000 2 1LI N-[(1s,2r)-3-{[1-(3-tert-butylphenyl)cyclohexyl]amino}-1-(3,5-difluorobenzyl)-2-hydroxypropyl]acetamide 0.919 3 1BL (2r)-5-{[(2s,3r)-4-{[1-(3-tert-butylphenyl)cyclohexyl]amino}-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]amino}-2-hydroxy-5-oxopentanoic acid 0.791 4 C6A N-[(2s,3r)-4-{[(2r,4s)-2-cyclopropyl-6-(2,2-dimethylpropyl)-3,4-dihydro-2h-chromen-4-yl]amino}-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]acetamide 0.738 5 842 N-[(1s,2r)-1-(3,5-difluorobenzyl)-2-hydroxy-3-({1-[3-(1h-pyrazol-1-yl)phenyl]cyclohexyl}amino)propyl]acetamide 0.714