1 21G (2s,3s)-3-[[5-fluoranyl-2-(5-fluoranyl-1h-pyrrolo[2,3-B]pyridin-3-yl)pyrimidin-4-yl]amino]bicyclo[2.2.2]octane-2-carboxylic acid 1.000 2 BYB (2~{S},3~{S})-3-[[5-fluoranyl-2-(5-fluoranyl-1~{H}-pyrazolo[3,4-B]pyridin-3-yl)pyrimidin-4-yl]amino]bicyclo[2.2.2]octane-2-carboxylic acid 0.933 3 KWN (1~{S},2~{S},3~{S},6~{R})-2-[[2-[5,7-bis(fluoranyl)-1~{H}-indol-3-yl]-5-fluoranyl-pyrimidin-4-yl]amino]-3,6-dimethyl-cyclohexane-1-carboxylic acid 0.788 4 4EW 2-(5-chloro-1h-pyrrolo[2,3-B]pyridin-3-yl)-5-fluoro-N-[(1r,2s,3s,4r)-3-(1h-tetrazol-5-yl)bicyclo[2.2.2]oct-2-yl]pyrimidin-4-amine 0.714