1 1BE N-(6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)-3-[2-propyl-4-(1h-pyrazol-4-yl)thiophen-3-yl]-L-alanine 1.000 2 1BF N-(6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)-3-[4-(1h-pyrazol-4-yl)thiophen-3-yl]-L-alanine 0.906 3 1B8 3-[2-bromo-4-(1h-pyrazol-4-yl)thiophen-3-yl]-N-(6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)-L-alanine 0.879 4 1BC 2-{(1s)-1-{[(1z)-6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1(2h)-ylidene]amino}-2-[2-propyl-4-(1h-pyrazol-4-yl)thiophen-3-yl]ethyl}pyrimidin-4(5h)-one 0.744 5 1B7 N-(6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)-3-(4-propylthiophen-3-yl)-L-alanine 0.735 6 1B9 3-(4-bromothiophen-3-yl)-N-(6-chloro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)-L-alanine 0.727