1 0N6 (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 1.000 2 1L4 N-[(2r)-3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-8-fluoro-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 0.969 3 1L8 8-fluoro-N-{(2r)-1-oxo-1-(pyrrolidin-1-yl)-3-[3-(trifluoromethyl)phenyl]propan-2-yl}-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide 0.857 4 FD3 N-alpha-(2-naphthylsulfonyl)-3-amidino-L-phenylalanine piperazide 0.829 5 FD1 N-alpha-(2-naphthylsulfonyl)-N-(3-amidino-L-phenylalaninyl)-D-pipecolinic acid 0.763 6 FD4 N-alpha-(2-naphthylsulfonyl)-N(3-amidino-L-phenylalaninyl)-4-acetyl-piperazine 0.763 7 FD2 N-alpha-(2-naphthylsulfonyl)-N(3-amidino-L-phenylalaninyl)isopipecolinic acid methyl ester 0.744 8 0ZG 3-[(2s)-2-{[(4-methylphenyl)sulfonyl]amino}-3-oxo-3-piperidin-1-ylpropyl]benzenecarboximidamide 0.743 9 730 (S)-3-(3-(4-(2-guanidinoethyl)piperidin-1-yl)-2-(naphthalene-2-sulfonamido)-3-oxopropyl)benzimidamide 0.707