1 0MP N-((2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-((6'-neopentyl-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-B]pyridin]-4'-yl)amino)butan-2-yl)acetamide 1.000 2 0KN (2r)-N-[(2s,3r)-1-(1,3-benzodioxol-5-yl)-4-{[(4'S)-6'-(2,2-dimethylpropyl)-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-B]pyridin]-4'-yl]amino}-3-hydroxybutan-2-yl]-2-methoxypropanamide 0.829 3 C6A N-[(2s,3r)-4-{[(2r,4s)-2-cyclopropyl-6-(2,2-dimethylpropyl)-3,4-dihydro-2h-chromen-4-yl]amino}-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]acetamide 0.821 4 0K9 (2r)-N-{(2s,3r)-4-{[(4'S)-6'-(2,2-dimethylpropyl)-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-B]pyridin]-4'-yl]amino}-3-hydroxy-1-[3-(1,3-thiazol-2-yl)phenyl]butan-2-yl}-2-methoxypropanamide 0.791 5 916 N-[(2s,3r)-4-{[(4s)-6-(2,2-dimethylpropyl)-2,2-dimethyl-3,4-dihydro-2h-thieno[2,3-B]pyran-4-yl]amino}-3-hydroxy-1-phenylbutan-2-yl]acetamide 0.763 6 1R8 (3s)-3-[(1r)-2-{[(4s)-6-ethyl-3,4-dihydrospiro[chromene-2,1'-cyclobutan]-4-yl]amino}-1-hydroxyethyl]-4-azabicyclo[10.3.1]hexadeca-1(16),12,14-trien-5-one 0.732 7 1QT (3s)-3-[(1r)-2-{[(4s)-6-ethyl-3,4-dihydrospiro[chromene-2,1'-cyclobutan]-4-yl]amino}-1-hydroxyethyl]-4-azabicyclo[11.3.1]heptadeca-1(17),13,15-trien-5-one 0.714